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@sigtrans-sttt.bsky.socialOct 17, 2026, 2:00 AM

Can targeting lipid metabolism improve treatment of SDH-deficient gastrointestinal stromal tumors? This phase 1b study reports promising activity of olverembatinib, which suppresses CD36 expression and lipid uptake.

#STTT #OpenAccess: doi.org/10.1038/s413...
#CancerMetabolism #LipidUptake

Olverembatinib, a multikinase inhibitor that modulates lipid metabolism, in advanced succinate dehydrogenase-deficient gastrointestinal stromal tumors: a phase 1b study and translational research
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